PK-ePD linear regression | IV AL | IV AS | |||||||
---|---|---|---|---|---|---|---|---|---|
Parameter | Analyte | a | b | r2 | p | a | b | rp | p |
Cmax (mM) | Parent | Â | Â | Â | Â | 1.04 | 7.45 | 0.807 | <0.001 |
t1/2 (min) | Parent | 0.69 | 7.89 | 0.964 | <0.001 | Â | Â | Â | Â |
Metabolite | Â | Â | Â | Â | 0.72 | 9.09 | 0.743 | 0.001 | |
AUC0–∞ (mM min) | Parent | 7.88 | 124 | 0.951 | <0.001 |  |  |  |  |
Combined | Â | Â | Â | Â | 1.12 | 265 | 0.847 | <0.001 | |
AUC0–20 (mM min) | Parent | 8.09 | 32.7 | 0.751 | 0.005 | 0.94 | 76.3 | 0.803 | <0.001 |